{"id":8445,"date":"2016-07-27T21:10:46","date_gmt":"2016-07-28T00:10:46","guid":{"rendered":"http:\/\/scienceblogs.com.br\/hypercubic\/?p=8445"},"modified":"2016-07-27T21:10:46","modified_gmt":"2016-07-28T00:10:46","slug":"na-cola-do-ebola","status":"publish","type":"post","link":"https:\/\/www.blogs.unicamp.br\/hypercubic\/2016\/07\/na-cola-do-ebola\/","title":{"rendered":"Na cola do Ebola"},"content":{"rendered":"<p align=\"justify\"><a href=\"http:\/\/scienceblogs.com.br\/hypercubic\/files\/2016\/07\/Ebola_Virus_HQ.jpg\" data-rel=\"lightbox-image-0\" data-rl_title=\"\" data-rl_caption=\"\"><img fetchpriority=\"high\" decoding=\"async\" style=\"float: none;padding-top: 0px;padding-left: 0px;margin-left: auto;padding-right: 0px;margin-right: auto;border: 0px\" title=\"\" src=\"http:\/\/scienceblogs.com.br\/hypercubic\/files\/2016\/07\/Ebola_Virus_HQ_thumb.jpg\" alt=\"Ebola_Virus_HQ\" width=\"692\" height=\"360\" border=\"0\" \/><\/a><\/p>\n<p align=\"justify\">A chave-de-fenda-s\u00f4nica do Doutor n\u00e3o funciona em madeira, o Super-Homem enfraquece diante da kriptonita, o Homem de Ferro tem problemas card\u00edacos, o Batman \u00e9 uma crian\u00e7a traumatizada e as teias do Homem-Aranha n\u00e3o s\u00e3o l\u00e1 muito \u00fateis longe dos arranha-c\u00e9us nova-iorquinos. No mundo dos v\u00edrus, o super-her\u00f3i \u00e9 o Ebola (EBOV), que tamb\u00e9m tem um ponto fraco.<!--more--><\/p>\n<p align=\"justify\">O problema, para n\u00f3s, \u00e9 que o ponto fraco do EBOV n\u00e3o \u00e9 t\u00e3o \u00f3bvio quanto o dos protagonistas das hist\u00f3rias em quadrinhos. H\u00e1 quarenta anos os cientistas lutam para encontrar o calcanhar de Aquiles desse vil\u00e3o implac\u00e1vel. Em 30 epis\u00f3dios, o Ebola j\u00e1 matou centenas de milhares de pessoas. Na \u00faltima epidemia \u2014 a mais grave, registrada na \u00c1frica Ocidental entre 2014 e 2015 \u2014, redobraram-se os esfor\u00e7os de pesquisa diante de uma ame\u00e7a potencialmente global.<\/p>\n<p align=\"justify\">Os resultados dessa maratona de pesquisas come\u00e7am a aparecer. Cientistas da Universidade de Oxford, no Reino Unido, encontraram uma poss\u00edvel vulnerabilidade do EBOV: seu bolso.<\/p>\n<p align=\"justify\"><a href=\"http:\/\/scienceblogs.com.br\/hypercubic\/files\/2016\/07\/Ebola-Zaire.jpg\" data-rel=\"lightbox-image-1\" data-rl_title=\"\" data-rl_caption=\"\"><img decoding=\"async\" style=\"float: none;padding-top: 0px;padding-left: 0px;margin-left: auto;padding-right: 0px;margin-right: auto;border: 0px\" title=\"\" src=\"http:\/\/scienceblogs.com.br\/hypercubic\/files\/2016\/07\/Ebola-Zaire_thumb.jpg\" alt=\"Ebola-Zaire\" width=\"1138\" height=\"598\" border=\"0\" \/><\/a><\/p>\n<p align=\"justify\">Como se pode ver acima, v\u00edrus nada mais s\u00e3o que um novelo min\u00fasculo de prote\u00ednas e material gen\u00e9tico, que s\u00f3 fazem estrago quando conseguem entrar dentro das c\u00e9lulas. Foi nessa etapa de entrada que os pesquisadores de Oxford buscaram pistas. O Ebola n\u00e3o tem um p\u00e9 para derrubar as portas das c\u00e9lulas, nem uma bazuca: usa uma esp\u00e9cie de cola chamada glicoprote\u00edna. Essa arma do EBOV j\u00e1 era conhecida, mas agora a glicoprote\u00edna p\u00f4de ser observada em alta resolu\u00e7\u00e3o.<\/p>\n<p align=\"justify\"><span style=\"font-family: Georgia;font-size: medium\"><strong>No bolso d\u00f3i mais<\/strong><\/span><\/p>\n<p align=\"justify\">Em artigo publicado em 07\/07 na <em>Nature<\/em>, Yuguang Zhao <em>et al.<\/em> descrevem os detalhes dessa glicoprote\u00edna, formada por duas sub-unidades \u2014 GP-1 e GP-2. Na cola do Ebola, os pesquisadores encontraram algo interessante: a jun\u00e7\u00e3o entre GP-1 e GP-2 n\u00e3o \u00e9 perfeita e \u00e9 a\u00ed que pode estar o ponto fraco do EBOV. Zhao e seus colegas observaram uma dobra ou bolso nessa jun\u00e7\u00e3o. O que aconteceria se esse bolso fosse preenchido?<\/p>\n<p align=\"justify\">Teoricamente, o preenchimento desse bolso afetaria o mecanismo de a\u00e7\u00e3o da glicoprote\u00edna, dificultando ou impedindo a entrada do EBOV numa c\u00e9lula. Surpreendentemente, os pesquisadores logo descobriram em testes feitos com ratos que esse bolso poderia ser preenchido com duas drogas j\u00e1 dispon\u00edveis no mercado. Uma \u00e9 o toremifeno, j\u00e1 usado em coquet\u00e9is de quimioterapia. A outra droga, por\u00e9m, \u00e9 ainda mais comum: trata-se do anti-inflamat\u00f3rio e analg\u00e9sico ibuprofeno.<\/p>\n<p align=\"justify\">As mol\u00e9culas desses dois medicamentos encaixaram-se no bolso da glicoprote\u00edna do v\u00edrus Ebola, neutralizando sua virul\u00eancia. Como j\u00e1 s\u00e3o drogas conhecidas e testadas em humanos, os cientistas v\u00e3o poder pular algumas etapas da pesquisa. Ainda assim mais estudos ser\u00e3o necess\u00e1rios. O pr\u00f3ximo passo \u00e9 tentar replicar esse efeito em macacos, que t\u00eam um sistema imune bem mais parecido com o nosso. Mesmo que esse tratamento n\u00e3o seja bem-sucedido em humanos, ele aponta um caminho promissor pois o Ebola tem um ponto fraco. S\u00f3 falta saber como coloc\u00e1-lo no bolso.<\/p>\n<p style=\"padding-left: 30px\" align=\"justify\"><strong><span style=\"font-family: Georgia;font-size: medium\">Refer\u00eancia<\/span><\/strong><\/p>\n<p style=\"padding-left: 30px\" align=\"justify\"><span style=\"font-family: Georgia\"><a href=\"http:\/\/scienceblogs.com.br\/hypercubic\/files\/2012\/07\/rb2_large_gray25.png\" data-rel=\"lightbox-image-2\" data-rl_title=\"\" data-rl_caption=\"\" title=\"\"><img decoding=\"async\" class=\"alignleft size-full wp-image-3123\" src=\"http:\/\/scienceblogs.com.br\/hypercubic\/files\/2012\/07\/rb2_large_gray25.png\" alt=\"rb2_large_gray25\" width=\"70\" height=\"85\" \/><\/a>Yuguang Zhao <em>et al.<\/em> <strong>Toremifene interacts with and destabilizes the Ebola virus glycoprotein<\/strong> [<strong><em>Toremifeno interage com e desestabiliza a glicoprote\u00edna do v\u00edrus Ebola<\/em><\/strong>]. <em>Nature<\/em> 535, 169\u2013172 (07 July 2016). <a href=\"http:\/\/www.nature.com\/nature\/journal\/v535\/n7610\/full\/nature18615.html\">DOI: 10.1038\/nature18615<\/a><\/span><\/p>\n","protected":false},"excerpt":{"rendered":"<p>A chave-de-fenda-s\u00f4nica do Doutor n\u00e3o funciona em madeira, o Super-Homem enfraquece diante da kriptonita, o Homem de Ferro tem problemas card\u00edacos, o Batman \u00e9 uma crian\u00e7a traumatizada e as teias do Homem-Aranha n\u00e3o s\u00e3o l\u00e1 muito \u00fateis longe dos arranha-c\u00e9us nova-iorquinos. No mundo dos v\u00edrus, o super-her\u00f3i \u00e9 o Ebola (EBOV), que tamb\u00e9m tem um [&hellip;]<\/p>\n","protected":false},"author":486,"featured_media":8449,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"_eb_attr":"","_monsterinsights_skip_tracking":false,"_monsterinsights_sitenote_active":false,"_monsterinsights_sitenote_note":"","_monsterinsights_sitenote_category":0,"material-hide-sections":[],"pgc_sgb_lightbox_settings":"","_vp_format_video_url":"","_vp_image_focal_point":[],"footnotes":""},"categories":[34,35,53,86,217,275,315],"tags":[801,1280,1711,1854,3188,3300,3433,3442],"class_list":["post-8445","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-biologia","category-bioquimica-biologia","category-ciencia","category-divulgacao-cientifica","category-microbiologia","category-quadrinhos","category-tirinhas","tag-bolso","tag-ebola","tag-glicoproteina","tag-ibuprofeno","tag-super-herois","tag-toremifeno","tag-viloes","tag-virologia"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.6 - 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